Linker Hydrophilicity Modulates the Anticancer Activity of RGD-Cryptophycin Conjugates.
Anselmi, Michele ; Borbély, Adina Noémi ; Figueras Agustí, Eduard ; Michalek, Carmela ; Kemker, Isabell ; Gentilucci, Luca ; Sewald, NorbertIn: Chemistry - A European Journal, Jg. 27 H. 3, S. 1015-10222021LC-ToF-ESI-MS Patterns of Hirsutinolide-like Sesquiterpenoids Present in the Elephantopus mollis Kunth Extract and Chemophenetic Significance of Its Chemical [...]
Bitchagno Mbahbou, Gabin Thierry ; Koffi, Jean Garba ; Simo, Ingrid Konga ; Kagho, Donald Ulrich K. ; Ngouela, Augustin Silvere ; Lenta, Bruno Ndjakou ; Sewald, NorbertIn: Molecules, Jg. 26 H. 162021Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery
Borbély, Adina Noémi ; Figueras Agustí, Eduard ; Martins, Ana ; Bodero, Lizeth ; Raposo Moreira Dias, Andre ; Lopez Rivas, Paula ; Pina, Arianna ; Arosio, Daniela ; Gallinari, Paola ; Frese, Marcel ; Steinkühler, Christian ; Gennari, Cesare ; Piarulli, Umberto ; Sewald, NorbertIn: ChemistryOpen, Jg. 8 H. 6, S. 737-7422019Synthesis and Biological Evaluation of RGD–Cryptophycin Conjugates for Targeted Drug Delivery
Borbély, Adina Noémi ; Figueras Agustí, Eduard ; Martins, Ana ; Esposito, Simone ; Auciello, Giulio ; Monteagudo, Edith ; Di Marco, Annalise ; Summa, Vincenzo ; Cordella, Paola ; Perego, Raffaella ; Kemker, Isabell ; Frese, Marcel ; Gallinari, Paola ; Steinkühler, Christian ; Sewald, NorbertIn: Pharmaceutics, Jg. 11 H. 42019Synthesis and Biological Characterization of Monomeric and Tetrameric RGD-Cryptophycin Conjugates.
Borbély, Adina Noémi ; Thoreau, Fabien ; Figueras Agustí, Eduard ; Kadri, Malika ; Coll, Jean-Luc ; Boturyn, Didier ; Sewald, NorbertIn: Chemistry - A European Journal, Jg. 26 H. 12, S. 2602-26052020Zum Cycloadditionsverhalten von 5-Azido-4-trifluormethyl-1,3-azolen
Burger, K. ; Höß, E. ; Geith, K. ; Riede, J. ; Bissinger, P. ; Sewald, NorbertIn: Z. Naturforsch. B: Chem. Sci., Jg. 45 H. 12, S. 1695-17081990Reaktionen 4,4-Bis(trifluormethyl)-substituierter Heterodiene mit Alkinen / Reactions of 4,4-Bis(trifluoromethyl) Substituted Heterodienes with Alkyne [...]
Burger, Klaus ; Sewald, Norbert ; Huber, Erasmus ; Ottlinger, RalphIn: Zeitschrift für Naturforschung B, Jg. 44 H. 10, S. 1298-13121989In Vivo Antitumor Activity of a Novel Acetazolamide-Cryptophycin Conjugate for the Treatment of Renal Cell Carcinomas
Cazzamalli, Samuele ; Figueras Agustí, Eduard ; Petho, Lilla ; Borbély, Adina Noémi ; Steinkuhler, Christian ; Neri, Dario ; Sewald, NorbertIn: ACS Omega, Jg. 3 H. 11, S. 14726-147312018An RGD helper sequence in CagL of Helicobacter pylori assists in interactions with integrins and injection of CagA
Conradi, Jens ; Tegtmeyer, Nicole ; Wozna, Marta ; Wißbrock, Marco ; Michalek, Carmela ; Gagell, Corinna ; Cover, Timothy L. ; Frank, Ronald ; Sewald, Norbert ; Backert, SteffenIn: Frontiers in Cellular and Infection Microbiology, Jg. 2, S. 70 ff.2012Einzelmolekülexperimente in der synthetischen Biologie: ein Ansatz für das Affinitätsranking DNA-bindender Peptide
Eckel, Rainer ; Wilking, Sven David ; Becker, Anke ; Sewald, Norbert ; Ros, Robert ; Anselmetti, DarioIn: Angewandte Chemie, Jg. 117 H. 25, S. 3989-39932005Single-molecule experiments in synthetic biology: an approach to the affinity ranking of DNA-binding peptides
Eckel, Rainer ; Wilking, Sven David ; Becker, Anke ; Sewald, Norbert ; Ros, Robert ; Anselmetti, DarioIn: Angewandte Chemie (Intl. Edition), Jg. 44 H. 25, S. 3921-39242005Octreotide Conjugates for Tumor Targeting and Imaging.
Figueras Agustí, Eduard ; Martins, Ana ; Borbély, Adina Noémi ; Le Joncour, Vadim ; Cordella, Paola ; Perego, Raffaella ; Modena, Daniela ; Pagani, Paolo ; Esposito, Simone ; Auciello, Giulio ; Frese, Marcel ; Gallinari, Paola ; Laakkonen, Pirjo ; Steinkuhler, Christian ; Sewald, NorbertIn: Pharmaceutics, Jg. 11 H. 52019Bifunctional Reagents for Formylglycine Conjugation: Pitfalls and Breakthroughs
Janson, Nils ; Krüger, Tobias ; Karsten, Lennard ; Boschanski, Mareile ; Dierks, Thomas ; Müller, Kristian ; Sewald, NorbertIn: ChemBioChem, Jg. 21 H. 24, S. 3580-35932020Antimicrobial Furoquinoline Alkaloids from Vepris lecomteana (Pierre) Cheek & T. Heller (Rutaceae)
Kouam, Ariane ; Bissoue, Achille ; Tcho, Alain ; Happi, Emmanuel ; Waffo, Alain ; Sewald, Norbert ; Wansi, JeanIn: Molecules, Jg. 23 H. 12018Targeted Enzyme Engineering Unveiled Unexpected Patterns of Halogenase Stabilization
Minges, Hannah ; Schnepel, Christian ; Boettcher, Dominique ; Weiss, Martin S. ; Sproß, Jens ; Bornscheuer, Uwe T. ; Sewald, NorbertIn: ChemCatChem, Jg. 12 H. 3, S. 818-8312020Prenylated Flavonoids and C-15 Isoprenoid Analogues with Antibacterial Properties from the Whole Plant of Imperata cylindrica (L.) Raeusch (Gramineae)
Nago, Romeo ; Nayim, Paul ; Mbaveng, Armelle ; Mpetga, James ; Bitchagno Mbahbou, Gabin Thierry ; Garandi, Badawe ; Tane, Pierre ; Lenta Ndjakou, Bruno ; Sewald, Norbert ; Tene, Mathieu ; Kuete, Victor ; Ngouela, AugustinIn: Molecules, Jg. 26 H. 162021